基本信息
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磷酸伯氨喹
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63-45-6
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磷酸伯喹;扑疟喹;磷酸伯氨喹啉;
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C15H21N3O.2H3PO4
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455.34
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Primaquine diphosphate
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200-560-8
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Primaquine diphosphate
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226.6oC
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205-206°C (dec.)(lit.)
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451.1oC at 760 mmHg
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急性毒性:大鼠口经LD50: 177 mg/kg;小鼠口经LD50:68 mg/kg;小鼠腹腔LD50: 105 mg/kg;鸟静脉LD50:19300 ug/kg; 繁殖:大鼠口经TDLo:600 mg/kgSEX/DURATION : female 8-13 day(s) after conception; 大鼠口经TDLo:480 mg/kgSEX/DURATION : female 6-15 day(s) after conception;致突变:沙门氏菌Mutation in microorganismsTEST SYSTEM:200 ug/plate;<SPAN lang=EN-US style="FONT-SIZE: 9pt; FONT-FAMILY: Arial; mso-font-kerning: 0pt; ms
详细信息
抗疟药,用于控制间日疟与三日疟的复发和恶性疟的传播